Meclofenoxate (Centrophenoxine) (51-68-3) wikiō
ʻO ka paukū Meclofenoxate (Centrophenoxine) Snāʻike
Product Name | Meclofenoxate (Centrophenoxine) (51-68-3) |
Hawaiian Name | ʻO Clophenoxate; Meclophenoxate; ʻO Clofenoxin; Makahiki; 2- (dimethylamino) ethyl 2- (4-chlorophenoxy) acetate |
Brand Name | N / A |
Kōpana Drug | Anti-Allergic agents, Antineoplastic agents, Antiparasitic Age |
Kāleka CAS | 51-68-3 |
InChIKey | XZTYGFHCIAKPGJ-UHFFFAOYSA-N |
hakakino F'Oula | C12H16ClNO3 |
hakakino Wʻewalu | 257.71 g / mole |
Monoisotopic Mass | 257.081871 g / mole |
ʻO ka paila | 345.941 ° C ma 760 mmHg |
Fkū hou Pʻo kaʻaila | N / A |
ʻO ka Halifa-Ola | 2-4 hola |
kala like 'ole | keʻokeʻo |
Solakino | Pākuʻi wai: 2.9 mg / mL |
Ska hoʻokele Tka mahana | -20 ° C |
Apaukū | Ua hoʻohana nui ʻo Centrophenoxine pauka i ka lāʻau nootropics a me ka meaʻai no ka meaʻai. |
ʻO ka ʻike meclofenoxate (Centrophenoxine)
ʻO Meclofenoxate (Centrophenoxine), i kūʻai ʻia ma lalo o ka inoa inoa ʻo Lucidril, ʻo ia kekahi o nā nootropics mua loa a i ʻike ʻia i kapa ʻia nā "akamai". ʻO ka nootropic i kaulana a mahalo ʻia nona i hōʻoiaʻiʻo iā ia iho no ma mua o ʻelima mau makahiki o ka hoʻohana ʻana a me ka hoʻokūkū koʻikoʻi hau lapaʻau.
Kuhi ʻia i ka 1959 e nā ʻepekema i ka French National Scientific Research Center ma ke ʻano he mālama no ka maʻi o Alzheimer, ʻaʻole i lawa nā kahe o ke koko i ka lolo, and a me ka hoʻokaʻawale ʻana i nā makahiki o ka makahiki, ua hoʻohana nui ʻia kēia lāʻau lapaʻau no ka mālama ʻana i nā pilikia pili i ka makahiki, e like me nā ʻano like ʻole. me ke Alzheimer a me ka panikala. Hoʻohana pū ia e nā poʻe olakino e hoʻoikaika i ka hoʻomanaʻo a me ka hana cognitive a hoʻomaikaʻi maikaʻi i nā olakino olakino holoʻokoʻa.
Ua hōʻike ʻia nā noiʻi i ka pauma centrophenoxine e lilo i mea hoʻomanaʻo hoʻomanaʻo hoʻomanaʻo a me ka anti-kahiko anti.
I loko oʻEulopa, ua kuhikuhi ʻia no ka mālama ʻana i nā hoʻomanaʻo o ka makahiki e pili ana i ka makahiki, akā ua loaʻa ia ma luna o ke counter a me kahi mea hoʻolako i ka papaʻaina i ka US a me Kanada, kahi mea e hoʻohana pinepine ʻia no kāna mau hoʻohui ʻoluʻolu.
He aha ia o Meclofenoxate (Centrophenoxine)?
Ua hoʻohana ʻia ʻo Centrophenoxine ma ke ʻano he meaʻaiʻai no kona mau pono e hoʻoikaika ai i ka hana.
ʻO Centrophenoxine ka hui ʻana o ʻelua mau huahana:
ʻO Dimethyl-aminoethanol (DMAE), he waiwai kūlohelohe i loaʻa i kekahi mau meaʻai (iʻa, ka wai kai a me nā mea liʻiliʻi i loko o ka lolo. He mea puna mai ia i ka choline a loaʻa nā hopena e hoʻoikaika ai ka lolo.
ʻO Parachlorphenoxyacetic acid (pCPA), kahi paʻi synthetic o nā lāʻau ulu o ka lāʻau i kapa ʻia ʻo "auxins".
ʻO DMAE ka mea hana nui i kēia lāʻau lapaʻau. ʻAʻole pololei ʻo DMAE i ka pale koko-lolo. Akā, i loko o ka centrophenoxine, hiki iā ia ke hele i ka hala o ka lolo-lolo a hoʻokomo maikaʻi i ka lolo
Hoʻokomo ʻia i ke kino, hoʻohele ʻia kahi hapa o ka centrophenoxine i ka DMAE a me ka pCPA i loko o ka ate. A laila hoʻohuli ʻia ka DMAE i ka choline, aʻo ka koena centrophenoxine e kū nei i ke kino holoʻokoʻa.
Nā pono Meclofenoxate (Centrophenoxine) i loaʻa
Hiki ke kōkua ʻo Centrophenoxine i ka hoʻoulu ʻana i ka maʻi maʻi.
Hiki ke kōkua ʻo Centrophenoxine i nā hōʻailona o ka dyskinesia tardive.
Hoʻonui ka Centrophenoxine i ka hoʻomanaʻo a me ka aʻo ʻana, hiki ke hoʻomaikaʻi i ka hoʻomanaʻo ʻana i nā mea maʻi dementia.
Ua hōʻike ʻia ʻo Centrophenoxine e hoʻomaikaʻi i ka hoʻokumu ʻana, mālama, a loaʻa hou i nā hoʻomanaʻo. E hoʻomaikaʻi ʻia ka hana hoʻomanaʻo ʻana inā loaʻa iā mākou nā kiʻekiʻe kiʻekiʻe o ka acetylcholine. Hōʻike i ka hoʻonui ʻana o Centrophenoxine i nā hana cholinergic i hoʻokahi, ʻo kekahi o nā mea i hana ʻia he choline, ma waena o nā phospholipids like ʻole.
Hoʻohui i nā Cognitive Function
Hiki ke hoʻohana ʻia ʻo Centrophenoxine e like me ka prodrug DMAE a ʻoiai he mea nui loa kēia, ʻoiai mea maikaʻi loa kēia molekue i ka hōʻemi ʻana i nā molekoleko ʻē aʻe i loko o ka lolo e hiki ai ke hōʻemi i ka hana hōʻemi ma nā hana cognitive. Me kēia mau molekala e hoʻokuʻu ʻia, hiki i ka poʻe ʻelemakule ke hoʻolōʻihi i ko lākou wā lohi a hoʻohuli i kekahi mau ʻaoʻao o ka wā kahiko.
ʻO Centrophenoxine ka anti-Aging a me Neuroprotective Properties
Ua hōʻike ʻia ʻo Centrophenoxine e hoʻonui i ke ola o nā kiʻi a hiki i 50%.
Hoʻonui ka Centrophenoxine i ka Mood a me ka Motivation, hiki iā ia ke kōkua i ka hōʻoluʻolu o ka hopohopo.
Ke hōʻike nei nā haʻawina holoholona i ka centrophenoxine he nui ka hopena anti-anxiety
Hoʻopilikena (Centrophenoxine) metabolism
Hoʻohana nui ʻia ʻo Centrophenoxine ma ka hoʻopuka a hoʻonui ʻana i nā hana o ka choline. ʻO Choline ka mea i hoʻomaka ai ka acetylcholine, kahi neurotransmitter koʻikoʻi a palena ʻole i pili pū me ka cognitive acuity, plasticity, a me ka hoʻomanaʻo. ʻAʻole maopopo ia pehea ka hoʻonui pinepine ʻana o ka centrophenoxine i nā pae o ka choline a me acetylcholine, akā ua manaʻo ʻia e hāʻule maoli paha i ka choline a i hoʻohuli ʻia i kahi phospholipid waena o ka wā i hoʻohana ʻia e hana i ka acetylcholine. Ka mea ʻole o ke ala, ʻo ia ka mea hiki ke cholinergic i mea e loaʻa ai ka centrophenoxine me kahi pototika nootropic ikaika.
I ka hoʻohui ʻana o ka hana acetylcholine, ʻike pū ʻia ka centrophenoxine i kahi ikaika neuro ikaika e hoʻoulu ai i ka hana o ka lolo ma o ka hoʻomaikaʻi ʻana i ke kūmole glucose a hoʻonui i ka piʻi o ka oxygen. Me ka hana ʻana, hana nui ka sentrophenoxine i ka hana o ka lolo i ka hana pono, no laila e hoʻomaikaʻi ai i ke kiko, ʻona, a me ke ʻano o nā manaʻo, e hoʻokuʻu aku ana i ka ʻohu ʻohu ʻohu. E like me ka nui o ka antiioxidant, ke kahili nei i nā mea hoʻopuka manuahi, e hoʻohemo i nā mea kinikini a komo i ka hoʻoponopono hou ʻana i nā puna i hoʻopau ʻia. ʻO ka mea hope loa, e hōʻole ana i ka ʻōpū o ka cognitive ma o ka hōʻemi ʻana a i ʻole ke hoʻopau ʻana i ka kūkulu ʻana o nā huahana mea ʻōpala metabolic i manaʻo ʻia he "pālule a waimaka."
ʻO nā hopena ʻaoʻao a me ka palekana Meclofenoxate (Centrophenoxine).
Hoʻomaopopo pinepine ʻia ʻo Centrophenoxine e palekana a me ka mea ʻole-mea iona. Ua hoʻohana ʻia no ia ma kahi o 50 mau makahiki me ka ʻole o nā ʻaoʻao koʻikoʻi nui i hōʻike ʻia.
Ua ʻōlelo ʻia he lāʻau hoʻomau like ʻole no ka poʻe olakino olakino a me ke senile e loaʻa ana i ka hoʻomanaʻo hoʻomanaʻo.
Eia nō naʻe, ua loaʻa kekahi mau mea hoʻohana i nā hopena ʻoluʻolu a me nā hopena liʻiliʻi, e komo pū ana i ka nausea, ka poʻo, ka pilikia o ka gastrointestinal, a me ka hiamoe ʻole.
ʻAʻole ʻōlelo ʻia ʻo Centrophenoxine no nā wahine hāpai ma muli o ka ʻike DMAE.
Hoʻopilikena (Centrophenoxine) papa ʻaʻa
Loaʻa ka Centrophenoxine ma luna o ke kahua i loko o nā kapoti i loaʻa ka 200-300 mg pākahi. ʻO nā hoʻokolohua haukapila i hoʻāʻo ai i ka hopena o nā centrophenoxine ma nā hana cognitive i hoʻohana i nā kaila o kēlā me kēia lā
1,200 mg i nā olakino ololi a me nā poho a hiki i ka 2,000 mg i nā maʻi maʻi dementia.
Hoʻoponopono
He ʻohi puna maikaʻi ʻo Centrophenoxine a hiki iā ʻoe ke ʻike i ka nui o ka puʻupuʻu nootropic - ʻo kekahi o nā mea maʻamau ka Noopept a me Racetams.
ʻO Centrophenoxine a me Aniracetam Stack
Eia kekahi laʻana o kahi pānaʻi centrophenoxine e loaʻa ai i ka aniracetam racetam kaulana e hoʻolako ai i ka hoʻomanaʻo ʻana, ke ʻano, ka ʻoluʻolu, a me ka hoʻohaʻahaʻa ʻana i ka hopohopo.
1-2x i kēlā me kēia lā
250 mg Centrophenoxine
750 mg Aniracetam
ʻO Centrophenoxine a me Noopept Stack
Eia kekahi laʻana o ka pānaehana centrophenoxine me Noopept, hiki i kēia mākeke ke hoʻomaikaʻi i ka hoʻomanaʻo a me ke aʻo ʻana, ʻoiai e hāʻawi ana i nā waiwai neuroprotective.
1-2x i kēlā me kēia lā
250 mg Centrophenoxine
20 mg Noopept
Reference:
- I ka hana o ka physicochemistry intracellular i loko o ka hōʻike genitative i ka wā o ka wā ʻelemakule a me ka hopena o ka centrophenoxine. He loiloi. Zs-Nagy I et al. ʻO Arch Gerontol Geriatr. (1989)
- ʻO ka lāʻau Cholinergic no ka diskinesia tardive antardikotik. Tammenmaa-Aho I, Asher R, Soares-Weiser K, Bergman H. Cochrane Database Syst Rev. 2018 Mar 19
- ʻO ka hana Cytotoxic o nā ʻākena alkylating i ke alo o centrophenoxine a me kāna huahana hydrolysis. Sladek NE. ʻO J Pharmacol Exp Ther. 1977 Dek
- ʻO ka potentiation o ka antitumor activity o cyclophosphamide e centrophenoxine. Kanzawa F, Hoshi A, Tsuda S, Kuretani K. Gan. 1972 ʻAukake
- Centrophenoxine: nā hopena i ka ulu ʻana o ka lolo mammalian. Nandy K et al. J Am Geriatr Soc. (1978)
- ʻO ka hopena ʻokoʻa o ka meclofenoxate ma ka nalowale o ka hoʻomanaʻo i ka pākeke. Marcer D et al. Ika waʻumea. (1977)
- Nootropics pauku centrophenoxine (meclofenoxate) pōmaikaʻi a me ka paʻa