ʻO ke kiʻi wikiwikiʻo Ralist Orlistat (96829-58-2)
Hōʻemi Orlistat kaola (96829-58-2)
Aia ʻo Raw Orlistat pauma i loko o ka papa o nā lāʻau i kapa ʻia he lipase inhibitors e hana ʻia ma ke ālai ʻana i ka omo ʻana o 25% o ka momona i loko o kahi pāʻina a hoʻohana ʻia no ka pohō kaumaha o nā mākua kaumaha, 18 makahiki a ʻoi paha, ke hoʻohana ʻia me kahi calorie hoʻemi a me papaʻai momona momona. ʻO Raw Orlistat pauka kahi lāʻau i hoʻolālā ʻia e mālama i ka momona. ʻO kāna hana mua ke pale nei i ka lawe ʻana o nā momona mai ka papaʻai kanaka, a laila e hoʻēmi nei i ka lawe ʻana o ka calory. Hana ka pauka Raw Orlistat ma ka pāpā ʻana i ka liprease pancreatic, kahi enzyme e wāwahi i nā triglycerides i loko o ka ʻōpū. Me ka ʻole o kēia enzyme, pale ʻia nā triglycerides mai ka papaʻai mai ka hydrolyzed ʻia i loko o nā waikawa momona momona a hiki ke hoʻopau ʻia. Hoʻohana ʻia ka Raw Orlistat pauka i nā poʻe kaona kaupaona i loaʻa i ke koko kiʻekiʻe, diabetes, high kolesterol, a i ʻole nā maʻi puʻuwai. ʻO ka maikaʻi o ka paukū Raw Orlistat i ka paipai ʻana i ka pohō kaumaha he definite akā akahai. Hōʻike ʻia nā ʻikepili i hōʻuluʻulu ʻia mai nā hoʻokolohua hoʻokolohua i hāʻawi ʻia ka poʻe i ka pauka Raw Orlistat me ka hoʻololi ʻana i ka nohona, e like me ka papaʻai a me ka hoʻoikaika kino, e nalowale ma kahi o 2-3 kilo (4.4-6.6 lb) ʻoi aku ma mua o ka poʻe i lawe ʻole i ka lāʻau i loko o hoʻokahi makahiki. Hoʻemi haʻahaʻa ʻo Raw Orlistat kaola i ke kahe o ke koko a ʻike ʻia e pale i ka hoʻomaka ʻana o ka maʻi diabetes 2, inā mai ka pohō kaumaha a i ʻole nā hopena ʻē aʻe. Hoʻoemi ia i ka hanana o ka maʻi kō II i ka poʻe obese a puni ka nui e like me ka hoʻololi o ka nohona.
ʻOhana Lahui Orlistat (96829-58-2) Hōʻike
Product Name | Hoʻolālāʻo Orlistat |
Hawaiian Name | Tetrahydrolipstatin, 1-((3-hexyl-4-oxo-2-oxetanyl)methyl)dodecyl-2-formamido-4-methylvalerate |
Brand Name | Alli, Xenical |
Kōpana Drug | nā mea hoʻopuka lipase |
Kāleka CAS | 96829-58-2 |
InChIKey | AHLBNYSZXLDEJQ-FWEHEUNISA-N |
hakakino F'Oula | C29H53NO5 |
hakakino Wʻewalu | 495.745 g / mole |
Monoisotopic Mass | 495.392 g / mole |
Hoʻolaha Pʻo kaʻaila | <50 ° C |
Fkū hou Pʻo kaʻaila | ʻAʻohe lā i loaʻa |
ʻO ka Halifa-Ola | Ma muli o kaʻikeʻole i kaʻikepili,ʻo ka hapalua o ke ola o ka Raw Orlistat ka paukū i hoʻohuiʻia ma keʻanoʻo 1 a hiki i nā hola 2. |
kala like 'ole | ʻO ka pauma |
Palekana | DMSO: 19 mg / mL |
pūnaewele Tka mahana | mālama kelepili. 2-8 ° C |
Apaukū | E hoʻohana i ka mālamaʻana i ka momona. |
Kohana Orlistat paukū (96829-58-2) Hōʻike
ʻO Raw Orlistat ka paukū i loko o ka papa o nā lāʻau i kapaʻia he mau'āpena lipase e hana ana ma ke kāohiʻana i ka hoʻonaʻauaoʻana o 25% o ka momona i kahi pāʻina a ua hoʻohanaʻia no ka poho kaumaha ma ka poʻe pakeke, 18 makahiki aʻoi aku, ke hoʻohanaʻia me ka kalo-kalo. ʻai kai momona.
ʻO Raw Orlistat ka paukū lāʻau i hoʻohanaʻia e mālama i ka momona. ʻO kāna hana mua ke kāohi i ka laweʻana o nā momona mai kaʻai kanaka, a laila e ho'ēmi ana i kaʻai caloric. Hoʻolālāʻo Orlistat ka lāʻau i ka hanaʻana i ka lipase pancreatic, he enzyme e hōʻoki iho i nā'āhua i ka'ōpū. Ma waho o kēia enzyme,ʻaʻohe mea e hoʻonāʻia ai ka meaʻaiʻole i ka wai i loko o nā momona momona liʻiliʻi a ua hoʻoneʻeʻoleʻia. Hoʻomaopopoʻia ka papa inoaʻo Raw Orlistat i ka nui o ka poʻe i hiki ke loaʻa ka nui o ke koko, diabetes, high cholesterol, a maʻi maʻi paha. ʻO ka pono o Raw Orlistat ka paukū i ka hoʻonuiʻana i ka pohō kaumahaʻo ia heʻano kūpono. Hōʻikeʻia nāʻikepili mai nā hōʻike hoʻokolohua e hāʻawiʻia nā kānaka i hāʻawiʻia iā Raw Orlistat ka paukū e pili ana i nā loli ola, e like me kaʻai a me ka hoʻolālā, e pili ana i nā 2-3 kilokilo (4.4-6.6 lb) ma mua o ka poʻeʻaʻole i hoʻohana i ka lāʻau lāʻau i kēlā me kēia makahiki. ʻO ka lauliana Orlistat paukū e hoʻohaʻahaʻa haʻahaʻa i ke kahe o ke koko a hōʻikeʻia e pale i ka hoʻomakaʻana o ka maʻi maʻamauʻo 2, inā paha mai ka poho kaumaha a iʻole nā hopena'ē aʻe. Hoʻoemiʻia ka hopena o ka maʻi diabetes II i nā kānaka āpau e like me ka nui o nāʻano o ka nohoʻana o ke ola.
Orlistat ka lehu (96829-58-2) Mechanism of Action
ʻO Orlistat pauma kahi ʻano lipase e kāohi ana i ka lāʻau pohō kaumaha a he mea loaʻa hydrated o lipostatin. Hoʻopau ka Orlistat me ke koho pono ʻana i ka lipase ʻōpū a me ka lipase pancreatic, ʻoiai ʻaʻohe hopena i nā ʻenemi digestive (e like me amylase, trypsin a me chymotrypsin) a ma ka phospholipase, ʻaʻole hoʻi e pili i ka lawe ʻana o nā huaʻaleʻale, protein a me phospholipids. ʻAʻole hoʻokomo ʻia kēia lāʻau lapaʻau ʻoiai ka gastrointestinal tract a he hopena hoʻi e kāohi i ka lipase. Hoʻopau ʻo Orlistat i nā enzymes e ka paʻa ʻana o ka covalent i ke koena serine ma nā pūnaewele hana o ka ʻōpū a me ka lipre pancreatic. Pale kēia i ka momona o ka meaʻai mai ka wāwahi ʻia ʻana i mau waikawa momona a me diacylglycerol, no laila ʻaʻole hiki ke komo, e hoʻoliʻiliʻi ana i ka ʻai a me ka mālama ʻana i ke kaumaha o ke kino. ʻAʻole pono e hoʻopili ʻia kēia lāʻau e ke kino holoʻokoʻa e hopena. ʻO ka hana ʻoihana lāʻau a Orlistat kaukaʻi hilinaʻi: kahi lāʻau lapaʻau o Orlistat (120mg / d, tid, lawe ʻia me nā pāʻina), hui pū ʻia me kahi papaʻai calorie haʻahaʻa, hiki ke hōʻemi i 30% o ka momona momona. I kahi noiʻi e hoʻohālikelike ana i nā mea manawaleʻa maʻamau a momona, ʻaʻole i lawe nui ʻia ʻo Orlistat e ke kino a he haʻahaʻa koko haʻahaʻa loa hoʻi. Ma hope o hoʻokahi mahele waha (ʻo ka 800mg ka nui loa), ʻo ke kaukā koko o Orlistat i nā hola 8 e hiki mai ana <5 ng / ml. ʻO ka maʻamau, ʻo kahi lāʻau lapaʻau o Orlistat e lawe liʻiliʻi ʻia e ke kino a ʻaʻole e hōʻiliʻili i kahi manawa pōkole. I kahi hoʻokolohua in vitro, ʻo ka helu paʻa paʻa o Orlistat me nā protein ʻē aʻe i ʻoi aku ma mua o 99% (ʻo nā protein i hoʻopaʻa ʻia ʻo lipoproteins a me albumin), a ʻo kāna helu paʻa me nā ʻulaʻula koko he haʻahaʻa loa.
ʻO ka maikaʻi o ka lālā o Paula (96829-58-2)
▪ Orlistat hoʻemi i ka nui o ke kino ma mua o 20% ma ka lilo o ka momona o ke kino
▪ Kōkua ʻo Orlista iā ʻoe e aʻo pehea e helu ai i nā calories
▪ Hāʻawi ʻo Orlista iā ʻoe i kahi ʻano maikaʻi
▪ Loaʻa nā hopena maikaʻi a Orlista i ka hilinaʻi a me ka hauʻoli i nā mea hoʻohana
▪ Hāʻawi ʻo Orlista i nā hopena hoʻomau lōʻihi
▪ Hoʻemi ʻo Orlista i ke koʻikoʻi o nā maʻi e like me ka haʻawewe, ka maʻi kō, atherosclerosis a
ka cholesterol.
Manaʻoʻiaʻo Orlistat paukū (96829-58-2) Hōʻike
ʻO ka lālā i manaʻoʻia o Orlistat ka paukū heʻekolu mau manawa o ka lā me kaʻaiʻana i ka momona (ʻoiai a hiki i ka hola 120 ma hope o kaʻaiʻana). ʻAʻole i hōʻikeʻia ma luna o 1 mgʻekolu manawa i ka lā e hāʻawi i kekahi pono hou aʻe.
Pono nā kānaka ma kahiʻai palekana kūpono, hoʻemiʻia kalola me nā 30% o nā calorie mai ka momona. Pono e hoʻokaʻawaleʻia ka waiwai o ka momona, ka waiʻahu, a me ka protein i nā lāʻaiʻekolu. Inā hāʻule kekahiʻai i ka manawa aiʻoleʻaʻohe momona, hiki ke hoʻokuʻuʻia ka nui o Orlistat ka pau.
Ma muli o ka Orlistat pauma i hōʻike ʻia e hōʻemi i ka omo ʻana o kekahi mau wikamina hiki ke hoʻoheheʻe ʻia me ka momona a me betacarotene, pono e ʻōlelo ʻia i ka poʻe e lawe i kahi multivitamin e loaʻa ana nā huamona momona e hōʻoia i ka pono o ka meaʻai. Ma kahi ʻē aʻe, pono e lawe i ka mea hoʻowali wikamina ma kahi o 2 mau hola ma mua a ma hope paha o ka lawelawe ʻana o Orlistat pauma, e like me ka wā moe.
Nā hopena o ka umauma Orlistat (96829-58-2)
He mea maʻamau kaʻikeʻana i nā hopena o Orlistat powder i ka manawa āu e hoʻohana ai. Hiki paha iāʻoe keʻike i kekahi o nā hopenaʻaoʻao aʻaʻole like paha ma hope o ka laweʻana i kekahi lāʻau'ē aʻe. ʻO ka hapa nui o nā hopena e hele mai me ka hoʻohanaʻana iā Orlistat ka paukū e pili ana i keʻano e hana ai ia i kāu'ōnaehana digestive. Hiki keʻano haʻahaʻa a hana mau lākou i ka manawa e hoʻomaka aiʻoe i ka lāʻau. Hanaʻia kekahi ma hope o ka laweʻana i kahiʻai momona momona. ʻO kaʻoluʻolu, hele ka hapanui o lākou ma muli o ka hoʻomauʻana i ka hoʻomauʻana a ma hope o ka hahaiʻana i ka meaʻai maikaʻi.
Eia nā hopenaʻaoʻao maʻamau:
▲ Heʻeha
▲ ʻO kaʻeha a me ka hōʻinoʻole o ka maʻi
▲ ʻO ka holoiʻana o ka hinu
▲ Nā momona momona
▲ Paheʻe kaʻiliʻili
▲ Paʻi hope
Ma waho aʻe, ināʻoe e hele i loko o kekahi o kēia mau hopena, e mālamaʻoe i keʻano he pilikia kūikawā a kāhea koke i ke kauka. O lākou;
▲ ʻO ka nui o kaʻehaʻeha e heleʻole.
▲ Hive aiʻole ka hoʻoulu nuiʻana
▲ Pahū
▲ Ke hoʻomaha iki